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         5-HT(5-Hydroxytryptamine,5-羥色胺)神經遞質主要分布于松果體和下丘腦,可參與食欲、體溫調節,情緒,心血管功能,內分泌和抑郁等生理功能的調節。5-HT通過激動不同的5-HT受體,可具有不同藥理作用,因此,5-HT受體拮抗劑成為藥物設計的研究熱點[1][2]。百靈威作為專業試劑供應商,提供多種5-HT受體拮抗劑,為您的科研助力加油!

      • 質量穩定,性價比高
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      產品編號

      中英文名稱

      CAS

      規格

      384285

      Granisetron hydrochloride, 98%, a serotonin 5-HT3 receptor antagonist

      鹽酸格拉司瓊, 98%, 5-HT3受體拮抗劑

      107007-99-8

      200 mg

      1 g

      283801

      Ketanserin, 99%, a specific 5-HT2A serotonin receptor antagonist

      凱他色林, 99%, 特異性的5-HT2A 5-羥色胺受體拮抗劑

      74050-98-9

      250 mg

      1 g

      185928

      Lamotrigine, 98%, Novel anticonvulsant drug for inhibition of 5-HT

      拉莫三嗪, 98%, 抑制5-羥色胺(5-HT)吸收

      84057-84-1

      1 g

      5 g

      574335

      Mirtazapine, 99%, 5-HT Receptor

      米爾塔扎平, 99%, 5-HT受體抑制劑

      85650-52-8

      100 mg

      496697

      Olanzapine, 99%, High affinity for 5-HT2 serotonin and D2 dopamine receptor antagonist

      奧氮平, 99%, 5-HT2D2受體高親和性拮抗劑

      132539-06-1

      1 g

      5 g

      977215

      Paliperidone, 99%, potent D2 and 5-HT2A antagonist

      帕潘立酮, 99%, 高效D25HT2A拮抗劑

      144598-75-4

      10 mg

      50 mg

      144809

      Sumatriptan succinate, 98%, 5-HT1 receptor agonist

      琥珀酸舒馬曲普坦, 98%, 5-HT1 受體激動劑

      103628-48-4

      100 mg

      500 mg

      522188

      Tropisetron monohydrochloride, 99%, 5-HT3 receptor antagonist and α7-nicotinic receptor agonist

      鹽酸托烷司瓊, 99%, 5-HT3受體拮抗劑和α7-煙堿受體激動劑

      105826-92-4

      1 g

      5 g

      186095

      Ziprasidone hydrochloride monohydrate, 99%, a novel and potent dopamine and serotonin (5-HT) receptor antagonist

      齊拉西酮鹽酸鹽一水合物, 99%, 有效的dopamine serotonin (5-HT) receptor的拮抗劑

      138982-67-9

      250 mg

      1 g

                       

                                             Figure1                                                                                      Figure2

      Figure1: Structure of Lamotrigine (185928)[1] 

      Figure2: Interactions of Lamotrigine(185928) with the binding pocket (subdomain IB)[1]

       References

      [1] Poureshghi F, Ghandforoushan P, Safarnejad A, et al. Interaction of an antiepileptic drug, lamotrigine with human serum albumin (HSA): Application of spectroscopic techniques and molecular modeling methods[J]. Journal of Photochemistry and Photobiology B: Biology, 2017, 166: 187-192.

      [2]Yatham L N, Beaulieu S, Schaffer A, et al. Optimal duration of risperidone or olanzapine adjunctive therapy to mood stabilizer following remission of a manic episode: A CANMAT randomized double-blind trial[J]. Molecular psychiatry, 2016, 21(8): 1050-1056.

       

      產品編號

      中英文名稱

      CAS

      包裝規格

      163651

      (+)-Bicuculline, 99.5%, GABAA antagonist

      (+)-荷包牡丹堿, 99.5%, GABAA 拮抗劑

      485-49-4

      25 mg

      100 mg

      240627

      Candesartan cilexetil, 98%, ATR antagonist

      坎地沙坦酯, 98%, ATR 拮抗劑

      145040-37-5

      50 mg

      100 mg

      500 mg

      410760

      Cyproterone acetate, 98%, an androgen receptor (AR) antagonist

      環丙孕酮醋酸鹽, 98%, 一種雄激素受體拮抗劑

      427-51-0

      50 mg

      250 mg

      1 g

      195685

      Leuprorelin acetate, 98%, an agonist at pituitary GnRH receptors

      醋酸亮丙瑞林, 98%, 一種垂體促性腺激素受體抑制劑

      74381-53-6

      5 mg

      25 mg

      408413

      Tropicamide, 99%, potent selective M4 antagonist

      托品酰胺, 99%, 有效選擇性M4拮抗劑

      1508-75-4

      10 g

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